Brexpiprazole | CAS 913611-97-9 | Probechem Biochemicals

Chemical Structure : Brexpiprazole

CAS No.: 913611-97-9

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Brexpiprazole (OPC-34712)

货号: PC-24453Not For Human Use, Lab Use Only.

Brexpiprazole (OPC-34712) is an atypical orally active antipsychotic agent and partial agonist of human 5-HT1A and dopamine D2L receptor with Ki of 0.12 nM and 0.3 nM, respectively.

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50 mg	￥780	In stock
100 mg	￥1180	In stock
250 mg	￥1980	In stock
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生物&药学活性

Brexpiprazole (OPC-34712) is an atypical orally active antipsychotic agent and partial agonist of human 5-HT1A and dopamine D2L receptor with Ki of 0.12 nM and 0.3 nM, respectively.
Brexpiprazole (OPC-34712) is also a 5-HT2A receptor antagonist with Ki of 0.47 nM.
Brexpiprazole also shows potent antagonist activity at human noradrenergic α1B (Ki=0.17 nM) and α2C receptors (Ki=0.59 nM).

物理化学性质&存储条件

分子量	433.57
分子式	C25H27N3O2S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	7-(4-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)butoxy)quinolin-2(1H)-one

参考文献

1. Ishima T, et al. Eur Neuropsychopharmacol. 2015 Apr;25(4):505-11.

2. Yoshimi N, et al. Eur Neuropsychopharmacol. 2015 Mar;25(3):356-64.

Brexpiprazole (OPC-34712)

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物理化学性质&存储条件

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Brexpiprazole (OPC-34712)

生物&药学活性

物理化学性质&存储条件

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