BRL-44408 maleate |CAS: 681806-46-2 Probechem Biochemicals

Chemical Structure : BRL-44408 maleate

CAS No.: 681806-46-2

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BRL-44408 maleate (BRL44408)

货号: PC-60703Not For Human Use, Lab Use Only.

BRL-44408 maleate is a potent, selective α2A-adrenoceptor antagonist with Ki of 1.7 nM, 80-fold selectivity over α2B-adrenergic receptors.

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生物&药学活性

BRL-44408 maleate is a potent, selective α2A-adrenoceptor antagonist with Ki of 1.7 nM, 80-fold selectivity over α2B-adrenergic receptors.
BRL-44408 maleate significantly increases stimulated noradrenaline release in rat locus coeruleus slices at 0.1-1 uM, significantly increases the electrically induced release in rats.

物理化学性质&存储条件

分子量	331.372
分子式	C17H21N3O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-[(4,5-Dihydro-1H-imidazol-2-yl)methyl]-2,3-dihydro-1-methyl-1H-isoindole maleate

参考文献

1. Kiss JP, et al. Brain Res. 1995 Mar 20;674(2):238-44.

2. Callado LF, et al. Eur J Pharmacol. 1999 Jan 29;366(1):35-9.

3. Young P, et al. Eur J Pharmacol. 1989 Sep 22;168(3):381-6.

BRL-44408 maleate (BRL44408)

生物&药学活性

物理化学性质&存储条件

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BRL-44408 maleate (BRL44408)

生物&药学活性

物理化学性质&存储条件

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