BRL-37344 sodium | β3AR agonist | Probechem Biochemicals

Chemical Structure : BRL-37344 sodium

CAS No.: 127299-93-8

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BRL-37344 sodium (BRL37344A)

货号: PC-62018Not For Human Use, Lab Use Only.

BRL-37344 sodium (BRL 37344A) is a potent and selective β3 adrenoceptor (β3AR) agonist with Ki of 287 nM.

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5 mg	￥2180	In stock
10 mg	￥3580	In stock
25 mg	￥5980	In stock
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100 mg		Get quote

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生物&药学活性

BRL-37344 sodium (BRL 37344A) is a potent and selective β3 adrenoceptor (β3AR) agonist with Ki of 287 nM.
BRL-37344 has weaker binding affinity for β1 and β2 receptors with Ki of 1750 and 1120 nM, respectively.
BRL-37344 is a potent agonist in brown adipocytes (EC50 = 3.3 +/- 0.8 nM) than in white adipocytes (EC50=5.7 nM) or colon (EC50=27.5 nM).
BRL-37344 stimulates fuel oxidation by soleus muscle in vitro.

物理化学性质&存储条件

分子量	385.82
分子式	C19H21NO4ClNa
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Rel-2-[4-[(2S)-2-[[(2S)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]phenoxy]-acetic acid, monosodium salt

参考文献

1. Arch JR, et al. Nature. 1984 May 10-16;309(5964):163-5.

2. Oriowo MA, et al. J Pharmacol Exp Ther. 1996 Apr;277(1):22-7.

3. Board M, et al. Eur J Pharmacol. 2000 Oct 6;406(1):33-40.

BRL-37344 sodium (BRL37344A)

生物&药学活性

物理化学性质&存储条件

参考文献

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BRL-37344 sodium (BRL37344A)

生物&药学活性

物理化学性质&存储条件

参考文献

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