BPR1M492

Chemical Structure : BPR1M492

加入收藏

货号: PC-27320Not For Human Use, Lab Use Only.

BPR1M492 is a potent, selective, fast-acting μ-opioid receptor (MOR) agonist with EC50 of 4 nM in FLIPR Ca2+ assays, Emax=92.7%.

规格	价格	库存	数量
25 mg		Get quote
50 mg		Get quote
100 mg		Get quote

获取报价单

* 请选择数量再加入购物车

or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

生物&药学活性

BPR1M492 is a potent, selective, fast-acting μ-opioid receptor (MOR) agonist with EC50 of 4 nM in FLIPR Ca2+ assays, Emax=92.7%.
BPR1M492 demonstrates potent in vivo antinociception at 0.027 mg/kg, offering rapid pain relief within 5 min of subcutaneous injection.
BPR1M492 produced markedly milder withdrawal symptoms than TRV130 in mice.

物理化学性质&存储条件

分子量	320.44
分子式	C21H24N2O
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1H-Indene-2-carboxamide, 2,3-dihydro-N-[[(3R)-1,2,3,4-tetrahydro-2-methyl-3-isoquinolinyl]methyl]-

参考文献

1. Po-Wei Chang, et al. J Med Chem. 2026 Jun 11;69(11):13222-13247.

BPR1M492

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

BPR1M492

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Get Quotation Now

* Indicates a Required FieldYour information is safe with us.