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首页-小分子抑制剂&激动剂-Tyrosine Kinase-c-Kit-BLU-808
BLU-808

Chemical Structure : BLU-808

CAS No.: 3041025-10-6

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BLU-808 (BLU808, BLU 808)

货号: PC-21781Not For Human Use, Lab Use Only.

BLU-808 (BLU808) is a potent and selective wt c-KIT inhibitor, inhibits the autophosphorylation of wild-type c-Kit with IC50 of 0.3 nM, inhibits Exon 11 KIT with an IC50 of 0.9 nM.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    BLU-808 (BLU808) is a potent and selective wt c-KIT inhibitor, inhibits the autophosphorylation of wild-type c-Kit with IC50 of 0.3 nM, inhibits Exon 11 KIT with an IC50 of 0.9 nM.
    BLU-808 potently inhibits c-KIT-dependent phosphorylation and proliferation with IC50 values in the sub-nanomolar and nanomolar range, respectively.

    物理化学性质&存储条件

    分子量 529.58
    分子式 C27H28FN9O2
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20°C 12 个月; 4°C 6 个月
    配置液
    -80°C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    N-(5-(2-Cyclopropyl-2H-tetrazol-5-yl)-4-fluoro-2-methylphenyl)-5-(1-(2-hydroxy-2-methylpropyl)-3-methyl-1H-pyrazol-4-yl)pyrazolo[1,5-a]pyridine-3-carboxamide

    参考文献

    1. Patent WO2025255219A1. WIPO (PCT). 2025-06-04.

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