BIBS-39 (BIBS 39) | Angiotensin receptor antagonist | Probechem Biochemicals

Chemical Structure : BIBS-39

CAS No.: 133085-33-3

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BIBS-39 (BIBS39, BIBS 39)

货号: PC-45692Not For Human Use, Lab Use Only.

BIBS-39 (BIBS 39) is a selective nonpeptide angiotensin II receptor antagonist with Ki of 29 nM and 480 nM for AT1 and AT2 respectively.

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5 mg	￥1280	In stock
10 mg	￥1980	In stock
25 mg	￥3580	In stock
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生物&药学活性

BIBS-39 (BIBS 39) is a selective nonpeptide angiotensin II receptor antagonist with Ki of 29 nM and 480 nM for AT1 and AT2 respectively.
BIBS-39 shows no high affinity for other receptors, shifts the AII concentration-contractile response curves in isolated rabbit aorta with pA2 of 8.14 and a slope of 1.06.
BIBS-39 shows effective antihypertensives in the model of the renal hypertensive rat.

物理化学性质&存储条件

分子量	524.6533
分子式	C32H36N4O3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	DMSO: ≥ 32 mg/mL
Chemical Name/SMILES	[1,1'-Biphenyl]-2-carboxylic acid, 4'-[[2-butyl-6-[[(cyclohexylamino)carbonyl]amino]-1H-benzimidazol-1-yl]methyl]-

参考文献

1. Zhang J, et al. Eur J Pharmacol. 1992 Jul 21;218(1):35-41.

BIBS-39 (BIBS39, BIBS 39)

生物&药学活性

物理化学性质&存储条件

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BIBS-39 (BIBS39, BIBS 39)

生物&药学活性

物理化学性质&存储条件

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