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首页-小分子抑制剂&激动剂-GPCR-Free Fatty Acid Receptor (FFAR)-AM-5262
AM-5262

Chemical Structure : AM-5262

CAS No.: 1222088-90-5

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AM-5262 (AM5262)

货号: PC-63042Not For Human Use, Lab Use Only.

AM-5262 is a potent full GPR40 (FFA1) agonist with EC50 of 81 nM.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    AM-5262 is a potent full GPR40 (FFA1) agonist with EC50 of 81 nM.
    AM-5262 shows improved rat PK profile and general selectivity profile, enhances glucose stimulated insulin secretion (mouse and human islets) and improves glucose homeostasis in vivo (OGTT in HF/STZ mice) when compared to AM-1638.

    物理化学性质&存储条件

    分子量 514.637
    分子式 C33H35FO4
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20 °C 12 个月; 4°C 6 个月
    配置液
    -80 °C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (1R,2R)-6'-((2-((R)-2,2-dimethylcyclopentyl)-2'-fluoro-5'-methoxy-[1,1'-biphenyl]-4-yl)methoxy)-2',3'-dihydrospiro[cyclopropane-1,1'-indene]-2-carboxylic acid

    参考文献

    1. Wang Y, et al. ACS Med Chem Lett. 2013 May 7;4(6):551-5.

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