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首页-小分子抑制剂&激动剂-Membrane Transporter/Ion Channel-Sodium Channel-AM-2099
AM-2099

Chemical Structure : AM-2099

CAS No.: 1443373-17-8

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AM-2099 (AM2099)

货号: PC-26470Not For Human Use, Lab Use Only.

AM-2099 is a potent, selective inhibitor of voltage-gated sodium channel NaV1.7 with IC50 of 0.16 uM (hNaV1.7), with no actiivity against hNaV1.5.

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5 mg ￥780 In stock
10 mg ￥1180 In stock
25 mg ￥1980 In stock
50 mg ￥3280 In stock
100 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

AM-2099 is a potent, selective inhibitor of voltage-gated sodium channel NaV1.7 with IC50 of 0.16 uM (hNaV1.7), with no actiivity against hNaV1.5.
AM-2099 exhibits good selectivity over a range of NaV isoforms.
AM-2099exhibits dose-dependent reduction of scratching behavior in a histamine-induced scratching model.

物理化学性质&存储条件

分子量 466.45
分子式 C19H13F3N4O3S2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

7-Quinazolinesulfonamide, 4-[2-methoxy-4-(trifluoromethyl)phenyl]-N-2-thiazolyl-

参考文献

1. Marx IE, et al. ACS Med Chem Lett. 2016 Sep 21;7(12):1062-1067.

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